| 货号 | 0820/5 |
| 供应商 | Tocris |
| 生物活性 | Selectiveδ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations. |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 计算分子量 | 691.87 |
| 分子式 | C38H53N5O7 |
| 可溶性/溶解性 | Soluble to 69.19 mg/ml in DMSO and to 1 mg/ml in water |
| CAS号 | 89352-67-0 |
| 序列号 | YXXFL (Modifications: Tyr-1 = N,N-diallyl-Tyr, X = Aib) |
| 参考文献 | Cohenet al (1996) Opioid agonist activity of ICI 174864 and its carboxypeptidase degradation product, LY281217. J.Pharmacol.Exp.Ther. 238 769. PMID: 2875170. Cowanet al (1985) Studies in vivo with ICI-174,864 and [D-Pen2,D-Pen5]-enkephalin. Neuropeptides 5 311. PMID: 2987731. Hirninget al (1985) Studies in vitro with ICI-174,864 [D-Pen2,D-Pen5]-enkephalin (DPDPE) and [D-Ala2,NMePhe4,Gly-ol]-enkephalin (DAGO). Neuropeptides 5 383. PMID: 2987739. Cottonet al (1984) ICI-174,864: a highly selective antagonist for the opioid δ receptor. Eur.J.Pharmacol. 97 331. PMID: 6323195. |