| 货号 | 1004/50 |
| 别名 | 5-(4-Chlorophenyl)-4-methyl-3-(1-(2 |
| 供应商 | Tocris |
| 生物活性 | A potent and highly selective D4 dopamine receptor antagonist, with Ki values of > 1700, 770 and 3.5 nM at cloned human D2, D3 and D4receptors. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >98 % |
| 计算分子量 | 417.38 |
| 分子式 | C23H25N2ClO.HCl |
| 可溶性/溶解性 | Soluble to 10 mM in DMSO |
| CAS号 | 156337-32-5 |
| 参考文献 | Rowleyet al (1997) 4-Heterocyclylpiperidines as selective high-affinity ligands at the human dopamine D4 receptor. J.Med.Chem. 40 2374. PMID: 9240352. Rowleyet al (1996) 5-(4-Chlorophenyl)-4-methyl-3-(1-(2-phenylethyl)piperidin-4-yl)isoxazole: a potent, selective antagonist at human cloned dopamine D4 receptors. J. Med. Chem. 39 1943. PMID: 8642551. |