| 货号 | 0180/50 |
| 别名 | (Z)-3-[(Aminoiminomethyl)thio]prop- |
| 供应商 | Tocris |
| 生物活性 | More potent than either GABA or muscimol as an agonist at low affinity GABAA receptors and is thus a useful ligand to investigate GABA receptors linked to benzodiazepine receptors. Also a GABAA-ρ receptor antagonist. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 计算分子量 | 244.24 |
| 分子式 | C4H6N2O2S.H2SO4 |
| 可溶性/溶解性 | Soluble to 10 mM in water |
| CAS号 | 92138-10-8 |
| 参考文献 | Johnston (1996) GABAC receptors: relatively simple transmitter-gated ion channels? TiPS 17 319. PMID: 8885697. Holden-Dye and Walker (1988) ZAPA, (Z)-3-[(aminoiminomethyl)thio]-2-propenoic acid hydrochloride, a potent agonist at GABA-receptors on the Ascaris muscle cell. Br.J.Pharmacol. 95 3. PMID: 2851353. Allanet al (1986) Isothiouronium compounds as γ-aminobutyric acid agonists. Br.J.Pharmacol. 88 379. PMID: 3015310. |