货号 | 4220/50 |
别名 | 2-[4-(2,3,6,7-Tetrahydro-2,6-dioxo- |
供应商 | Tocris |
生物活性 | Adenosine receptor antagonist (Ki values are 42, 68 and 1130 nM for A1, A2B and A2Areceptors). |
运输条件 | Blue Ice |
存放说明 | Ambient |
纯度 | >98 % |
计算分子量 | 386.4 |
分子式 | C19H22N4O5 |
可溶性/溶解性 | Soluble to 50 mM in DMSO |
参考文献 | Thummler and Dunwiddie (2000) Adenosine receptor antagonists induce persistent bursting in the rat hippocampal CA3 region via an NMDA receptor-dependent mechanism. J.Neurophysiol. 83 1787. PMID: 10758091. Sebastiaoet al (1990) The inhibitory adenosine receptor at the neuromuscular junction and hippocampus of the rat: antagonism by 1,3,8-substituted xanthines. Br.J.Pharmacol. 101 453. PMID: 2257444. Jarviset al (1989) Autoradiographic characterization of high-affinity adenosine A2 receptors in the rat brain. Brain Res. 484 111. PMID: 2713675. |