货号 | 3761/50 |
别名 | 2-[(1R)-3-[Bis(1-methylethyl)amino] |
供应商 | Tocris |
生物活性 | High affinity muscarinic receptor antagonist (Ki = 3.3 nM). Active at all muscarinic receptor subtypes (M1 - M5); exhibits a greater effect on the bladder than salivary glands in vivo. |
运输条件 | Blue Ice |
存放说明 | 4℃ |
纯度 | >99 % |
计算分子量 | 475.57 |
分子式 | C22H31NO.C4H6O6 |
可溶性/溶解性 | Soluble to 10 mM in water and to 100 mM in DMSO |
CAS号 | 124937-52-6 |
参考文献 | Nilvebrant (2001) Clinical experiences with tolterodine. Life Sci. 68 2549. PMID: 11392625. Nilvebrantet al (1997) Tolterodine - a new bladder-selective antimuscarinic agent. Eur.J.Pharmacol. 327 195. PMID: 9200560. |