TC-T 6000 (50 MG)
货号:
5100/50 基本售价:
7961.3 元 规格:
50 mg
产品信息
概述货号 | 5100/50 |
别名 | 2,2'-[[4,8-Bis[bis(2-methylpropyl)amino]pyrimido[5,4-d]pyrimidine-2,6-diyl]diimino]bis-ethanol |
性能供应商 | Tocris |
生物活性 | Potent equilibrative nucleoside transporter 4 (ENT4) inhibitor (IC50 = 74.4 nM). Exhibits 20-fold and 80-fold selectivity for ENT4 over ENT2 and ENT1, respectively. |
运输条件 | Blue Ice |
存放说明 | Ambient |
纯度 | >98 % |
计算分子量 | 504.71 |
分子式 | C26H48N8O2 |
可溶性/溶解性 | Soluble to 20 mM in DMSO and to 20 mM in ethanol |
参考文献 | Wanget al (2013) Dipyridamole analogs as pharmacological inhibitors of equilibrative nucleoside transporters. Identification of novel potent and selective inhibitors of the adenosine transporter function of human equilibrative nucleoside transporter 4 (hENT4). Biochem.Pharmacol. 86 1531. PMID: 24021350. |