货号 | 0384/50 |
供应商 | Tocris |
生物活性 | Very potent inhibitor of cathepsin L (Ki = 0.6 nM) and the strongest inhibitor of cathepsin B (Ki = 100 nM) amongst the peptide aldehydes. Also inhibits processing of malaria aspartic hemoglobinases plasmepsins I and II in vitro. |
运输条件 | Blue Ice |
存放说明 | -20℃ |
计算分子量 | 401.56 |
分子式 | C19H35N3O4S |
可溶性/溶解性 | Soluble to 10 mM in ethanol and to 100 mM in DMSO |
CAS号 | 136632-32-1 |
参考文献 | Franciset al (1997) Biosynthesis and maturation of the malaria aspartic hemogloninases plasmepsins I and II. J.Biol.Chem. 272 14961. PMID: 9169469. Sasakiet al (1990) Inhibitory effect of di- and tripeptidyl aldehydes on calpains and cathepsins. J.Enzyme Inhib. 3 195. PMID: 2079636. |