| 货号 | 5387/50 |
| 别名 | 1-Methyl-5-nitro-3-phenyl-1H-indole |
| 供应商 | Tocris |
| 生物活性 | Selective PAR4 antagonist (IC50 = 140 nM). Exhibits 70-fold selectivity for PAR4 over PAR1. |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 纯度 | >98 % |
| 计算分子量 | 282.29 |
| 分子式 | C16H14N2O3 |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO |
| 参考文献 | Wenet al (2014) Substituted indoles as selective protease activated receptor 4 (PAR4) antagonists: Discovery and SAR of ML354. Bioorg.Med.Chem.Lett. 24 4708. PMID: 25176330. |