货号 | 2759/50 |
别名 | 5,6,7,8-Tetrahydro-6-(2-propen-1-yl |
供应商 | Tocris |
生物活性 | Dopamine D2 receptor agonist, α2-adrenoceptor agonist and 5-HT3 receptor antagonist. Displays antiParkinsonian activity. |
运输条件 | Blue Ice |
存放说明 | Ambient |
纯度 | >98 % |
计算分子量 | 282.23 |
分子式 | C10H15N3S.2HCl |
可溶性/溶解性 | Soluble to 100 mM in water and to 100 mM in DMSO |
CAS号 | 36085-73-1 |
参考文献 | Maina and Mathews (2010) A functional fast scan cyclic voltammetry assay to characterize dopamine D2 and D3 autoreceptors in the mouse striatum. ACS Chem.Neurosci. 1 450. PMID: 20567609. Ricci and Taira (1999) Adrenoceptor involvement in the cardiovascular responses to B-HT 920 in sinoaortic denervated rats. Gen.Pharmacol. 32 29. PMID: 9888250. Nishioet al (1996) 5-HT3 receptor blocking properties of the antiParkinsonian agent, talipexole. Gen.Pharmacol. 27 779. PMID: 8842679. Robertsonet al (1993) In vivo comparisons of the effects of quinpirole and the putative presynaptic dopaminergic agonists B-HT 920 and SND 919 on striatal dopamine and acetylcholine release. J.Pharmacol.Exp.Ther. 264 1344. PMID: 8095550. |