| 货号 | 0740/50 |
| 别名 | 17-(Cyclopropylmethyl)-6,7-dehydro- |
| 供应商 | Tocris |
| 生物活性 | Highly selective non-peptide δ opioid antagonist, showing 223- and 346-fold greater activity at δ than at μ |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >99 % |
| 计算分子量 | 450.96 |
| 分子式 | C26H26N2O3.HCl |
| 可溶性/溶解性 | Soluble to 25 mM in water and to 100 mM in DMSO |
| CAS号 | 111469-81-9 |
| 参考文献 | Shippenberg and Heidbreder (1995) The δ-opioid receptor antagonist naltrindole prevents sensitization to the conditioned rewarding effects of cocaine. Eur.J.Pharmacol. 280 55. PMID: 7498254. Ossipovet al (1994) Naltrindole, an opioid δ antagonist, blocks the enhancement of morphine-antinociception induced by a CCKB antagonist in the rat. Neurosci. Lett. 181 9. PMID: 7898778. Portogheseet al (1990) Design of peptidomimetic δ opioid receptor antagonists using the message-address concept. J.Med.Chem. 33 1714. PMID: 2160538. |