TC-DAPK 6 (50 MG)
货号：
4301/50 基本售价：
6622.9 元 规格：
50 mg
产品信息
概述| 货号 | 4301/50 |
| 别名 | (4Z)-2-[(E)-2-Phenylethenyl)-4-(3-pyridinylmethylene)-5(4H)-oxazolone |
性能| 供应商 | Tocris |
| 生物活性 | Potent and selective, ATP-competitive inhibitor of death-associated protein kinase 1 (DAPK1) (IC50 values are 69 and 225 nM for DAPK1 and DAPK3 respectively, when assayed with 10 μM ATP). Displays selectivity for DAPK1 over a range of 48 other kinases, including Abl, AMPK, Chk1, Met and Src (IC50 > 10 μM). |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >98 % |
| 计算分子量 | 276.29 |
| 分子式 | C17H12N2O2 |
| 可溶性/溶解性 | Soluble to 50 mM in DMSO |
| 参考文献 | Okamotoet al (2009) Identification of death-associated protein kinases inhibitors using structure-based virtual screening. J.Med.Chem. 52 7323. PMID: 19877644. |
