PRMT4/CARM1 Inhibitor
货号：
11033-5mg 基本售价：
6370.0 元 规格：
5 mg
产品信息
概述| 货号 | 11033-5mg |
| 描述 | PRMT4/CARM1 Inhibitor selectively blocks the activity of PRMT4/CARM1 with an IC50 value of 7.1 µM.1 It displays very low affinity towards PRMT1 and SET7 with IC50 values of 63 and 943 µM, respectively.1 In human prostate cancer LNCaP cells, this compound reduced the prostate-specific antigen promoter activity at 8-10 µM.1 |
| 别名 | Protein Arginine Methyltransferase 4/Coactivator-Associated Arginine Methyltransferase 1 Inhibitor; |
性能| 供应商 | Cayman |
| 应用文献 |
1.Cheng, D.,Valente, S.,Castellano, S., et al. Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as coactivator-associated arginine methyltransferase 1 inhibitors: Enzyme selectivity and cellular activity. J. Med. Chem. 54(13), 4982-4932 (2011).
|
| 运输条件 | Wet ice in continental US; may vary elsewhere |
| 存放说明 | -20 |
| 纯度 | ≥95% |
| 计算分子量 | 555.3 |
| 分子式 | C26H21Br2NO3 |
| CAS号 | 1020399-49-8 |
| 稳定性 | ≥ 2 years |
声明| 本官网所有报价均为常温或者蓝冰运输价格，如有产品需要干冰运输，需另外加收干冰运输费。 |
