Bufuralol (hydrochloride)
货号：
17794-10mg 基本售价：
5824.0 元 规格：
10 mg
产品信息
概述| 货号 | 17794-10mg |
| 描述 | Bufuralol is a non-specific β-adrenergic blocker with affinity for both β1 and β2-adrenergic receptors. It acts as a potent β-adrenoceptor antagonist with partial agonist activity.1 It is primarily metabolized by cytochrome P450 (CYP) isoform CYP2D6, with CYP1A2 and CYP2C19 also contributing to 1’-hydroxylation.2 |
| 别名 | Ro 3-4787; |
性能| 供应商 | Cayman |
| 应用文献 |
1.Pringle, T.H.,Francis, R.J.,East, P.B., et al. Pharmacodynamic and pharmacokinetic studies on bufuralol in man. Br.J.Clin.Pharmac. 22, 527-534 (1986).
2.Narimatsu, S.,Takemi, C.,Kuramoto, S., et al. Stereoselectivity in the oxidation of bufuralol, a chiral substrate, by human cytochrome P450s. Chirality 15(4), 333-339 (2003).
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| 运输条件 | Room temperature in continental US; may vary elsewhere |
| 存放说明 | -20 |
| 纯度 | ≥95% |
| 计算分子量 | 297.8 |
| 分子式 | C16H23NO2 • HCl |
| CAS号 | 60398-91-6 |
| 稳定性 | ≥ 2 years |
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