| 货号 | 1797/25 |
| 别名 | (9Z)-N-[1-((R)-4-Hydroxbenzyl)-2-hy |
| 供应商 | Tocris |
| 生物活性 | Metabolically stable inhibitor of anandamide cellular uptake (Ki = 3 μM). Displays relatively low affinity for CB1 and CB2 receptors (Ki values are 5.1 and > 10 μM) and for vanilloid VR1 receptors (EC50 = 10 μM). Has minimal activity against FAAH (Ki > 50 μM). Active in vivo. |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >99 % |
| 计算分子量 | 431.66 |
| 分子式 | C27H45NO3 |
| 可溶性/溶解性 | Soluble to 10 mM in ethanol and to 10 mM in DMSO |
| 参考文献 | de Lagoet al (2004) In vivo pharmacological actions of two novel inhibitors of anandamide cellular uptake. Eur.J.Pharmacol. 484 249. PMID: 14744610. Ortaret al (2003) Novel selective and metabolically stable inhibitors of anandamide cellular uptake. Biochem.Pharmacol. 35 1473. PMID: 12732359. |