货号 | 1669/1 |
供应商 | Tocris |
生物活性 | Potent and selective tachykinin NK1 receptor agonist (EC50 = 2 nM in guinea pig vas deferens). Active in vivo. |
运输条件 | Blue Ice |
存放说明 | -20℃ |
计算分子量 | 766.01 |
分子式 | C40H59N7O6S |
可溶性/溶解性 | Soluble to 1 mg/ml in water |
CAS号 | 133156-06-6 |
序列号 | FFPLM (Modifications: Phe-1 = delta-Aminovaleryl-Phe, Leu-4 = (methyl)Leu, Met-5 = C-terminal amide) |
参考文献 | Sakuradaet al (1999) Spinal actions of GR73632, a novel tachykinin NK1 receptor agonist. Peptides 20 301. PMID: 10422886. Meiniet al (1995) GR 73,632 and [glu(OBzl)11]substance P are selective agonists for the septide-sensitive tachykinin NK1 receptor in the rat urinary bladder. Neuropeptides 28 99. PMID: 7538205. Hall and Morton (1991) Novel ligands confirm NK-1 receptor-mediated modulation of neurotransmission in the guinea pig vas deferens preparation. Ann.N.Y.Acad.Sci. 632 404. PMID: 1719888. |