| 货号 | 1663/10 |
| 别名 | 4-[(αR*)-α-((2S*,5R*)-4-Allyl-2,5-dim |
| 供应商 | Tocris |
| 生物活性 | Potent, selective non-peptide δ-opioid receptor agonist. Ki values are 1.8, 15 and 34 nM for δ,μandκ receptors respectively. Centrally active following systemic administration in vivo. |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >99 % |
| 计算分子量 | 435.61 |
| 分子式 | C27H37N3O2 |
| 可溶性/溶解性 | Soluble to 100 mM in 1eq. HCl |
| CAS号 | 155836-52-5 |
| 参考文献 | Broomet al (2002) Comparison of receptor mechanisms and efficacy requirements for δ-agonist-induced convulsive activity and antinociception in mice. J.Pharmacol.Exp.Ther. 303 723. PMID: 12388657. Changet al (1993) A novel, potent and selective nonpeptidic delta opioid receptor agonist BW373U86. J.Pharmacol.Exp.Ther. 267 852. PMID: 8246159. Dykstraet al (1993) A novel delta opioid agonist, BW373U86, in squirrel monkeys responding under a schedule of shock titration. J.Pharmacol.Exp.Ther. 267 875. PMID: 8246162. |