(R)-MG 132 ( )
货号：
6033/10 基本售价：
4094.7 元 规格：
10 mg
产品信息
概述| 货号 | 6033/10 |
| 别名 | N-[(Phenylmethoxy)carbonyl]-L-leucyl-N-[(1S)-1-formyl-3-methylbutyl]-D-leucinamide |
性能| 供应商 | Tocris |
| 生物活性 | Potent 20S proteasome inhibitor (IC50 = 0.22 nM). Exhibits cytostatic and cytotoxic effects in tumor cells in vitro. |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 纯度 | >98 % |
| 计算分子量 | 475.63 |
| 分子式 | C26H41N3O5 |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO and to 20 mM in ethanol |
| 参考文献 | Mroczkiewiczet al (2010) Studies of the synthesis of all stereoisomers of MG-132 proteasome inhibitors in the tumor targeting approach. J.Med.Chem. 53 1509. PMID: 20112914. |
