ML 18 (10 MG)
货号:
5599/10 基本售价:
4005.4 元 规格:
10 mg
产品信息
概述货号 | 5599/10 |
别名 | (αS)-N-[[1-(4-Methoxyphenyl)cyclohexyl]methyl-α-[[[(4-nitrophenyl)amino]carbonyl]amino]-1H-indole-3-propanamide |
性能供应商 | Tocris |
生物活性 | Bombesin receptor subtype 3 (BRS-3) antagonist (IC50 = 4.8 μM). Also binds GRPR (IC50 = 16 μM). Inhibits BA1-stimulated cytosolic Ca2+ and suppresses cell proliferation in a lung cancer model in vitro. |
运输条件 | Blue Ice |
存放说明 | -20℃ |
纯度 | >98 % |
计算分子量 | 569.65 |
分子式 | C32H35N5O5 |
可溶性/溶解性 | Soluble to 100 mM in DMSO |
参考文献 | Moodyet al (2015) ML-18 is a non-peptide bombesin receptor subtype-3 antagonist which inhibits lung cancer growth. Peptides 64 55. PMID: 25554218. |