| 货号 | 1818/1 |
| 供应商 | Tocris |
| 生物活性 | Peptide agonist for sst2, sst3 and sst5 somatostatin receptors. IC50/Kd values (nM) at cloned human somatostatin receptors are: 290 - 1140 (sst1), 0.4 - 2.1 (sst2), 4.4 - 34.5 (sst3), > 1000 (sst4), and 5.6 - 32 (sst5). |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 计算分子量 | 1019.24 |
| 分子式 | C49H66N10O10S2 |
| 可溶性/溶解性 | Soluble to 1.20 mg/ml in water |
| CAS号 | 79517-01-4 |
| 序列号 | FCFWKTCT (Modifications: Phe-1 = D-Phe, Trp-4 = D-Trp, Thr-8 = Thr-ol, Disulfide bridge between 1 - 7) |
| 参考文献 | Hannonet al (2002) Drug design at peptide receptors. Somatostatin receptor ligands. J.Mol.Neurosci. 1815. Hoyeret al (1994) Molecular pharmacology of somatostatin receptors. Naunyn Schmiedebergs Arch.Pharmacol. 350 441. PMID: 7870182. Raynoret al (1993) Cloned somatostatin receptors: identification of subtype-selective peptides and demonstration of high affinity binding to linear peptides. Mol.Pharmacol. 43 838. PMID: 8100350. |