| 货号 | 4919/1 |
| 供应商 | Tocris |
| 生物活性 | SelectivehMC3 receptor antagonist (IC50 = 210 nM). Exhibits no activity at hMC4 receptors and hMC5receptors. |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 计算分子量 | 1008.19 |
| 分子式 | C51H69N13O9< |
| 可溶性/溶解性 | Soluble to 1 mg/ml in 25% ethanol / water |
| 序列号 | XDXXRWK (Modifications: X-1 = Ac-Nle, X-3 = beta-Ala, X-4 = D-2-Nal, Lys-7 = C-terminal amide, Asp-2, Lys-7, Cyclized) |
| 参考文献 | Griecoet al (2007) Further structure-activity studies of lactam derivatives of MT-II and SHU-9119: their activity and selectivity at human melanocortin receptors 3, 4, and 5. Peptides. 28 1191. PMID: 17482720. |