| 货号 | 1699/50 |
| 别名 | 9-Chloro-2-(2-furanyl)-[1,2,4]triaz |
| 供应商 | Tocris |
| 生物活性 | Potent adenosine receptor antagonist (Ki values are 3.5, 4.2, 16 and 51 nM for human A1, A2A, A2B and A3 receptors respectively). Orally active in vivo. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >99 % |
| 计算分子量 | 285.69 |
| 分子式 | C13H8ClN5O |
| 可溶性/溶解性 | Soluble to 5 mM in DMSO |
| CAS号 | 104615-18-1 |
| 参考文献 | Klotz (2000) Adenosine receptors and their ligands. Naunyn Schmiedebergs Arch.Pharmacol. 362 382. PMID: 11111832. Ghaiet al (1987) Pharmacological characterization of CGS 15943A: a novel nonxanthine adenosine antagonist. J.Pharmacol.Exp.Ther. 242 784. PMID: 3656113. Williamset al (1987) Biochemical characterization of the triazoloquinazoline CGS 15943, a novel, non-xanthine adenosine antagonist. J.Pharmacol.Exp.Ther. 241 415. PMID: 2883298. |