| 货号 | 1134/50 |
| 别名 | 4-[3-[(1,1-Dimethylethyl)amino]2-hy |
| 供应商 | Tocris |
| 生物活性 | Partial agonist at β3-adrenoceptors.β1- and β2-adrenoceptor antagonist (Ki values are 0.9, 4 and 88 nM for β1,β2andβ3 receptors respectively). |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 计算分子量 | 315.8 |
| 分子式 | C14H21N3O3.HCl |
| 可溶性/溶解性 | Soluble to 50 mM in water |
| CAS号 | 81047-99-6 |
| 参考文献 | Galitzkyet al (1998) On the presence of a putative fourth β-adrenoceptor in human adipose tissue. TiPS 19 164. PMID: 9652187. Preitneret al (1998) Metabolic response to various β-adrenoceptor agonists in β3-adrenoceptor knockout mice: evidence for a new β-adrenergic receptor in brown adipose tissue. Br.J.Pharmacol. 124 1684. PMID: 9756384. Strosberg and Pietri-Rouxel (1996) Function and regulation of the β3-adrenoceptor. TiPS 17 373. PMID: 8979772. Staehelinet al (1983) CGP-12177. A hydrophilic beta-adrenergic receptor radioligand reveals high affinity binding of agonists to intact cells. J.Biol.Chem. 258 3496. PMID: 6131886. |