货号 | 0475/100 |
别名 | 9,10-Dihydro-12'-hydroxy-2'-methyl-5'- |
供应商 | Tocris |
生物活性 | Partialα-adrenergic agonist. Partial D2 dopaminergic receptor agonist. Competitive 5-HT antagonist. |
运输条件 | Blue Ice |
存放说明 | Ambient |
纯度 | >98 % |
计算分子量 | 679.79 |
分子式 | C33H37N5O5CH3SO3H |
可溶性/溶解性 | Soluble to 100 mM in DMSO |
CAS号 | 6190-39-2 |
参考文献 | Lesageet al (1998) Agonistic properties of alniditan, sumatriptan and dihydroergotamine on human 5-HT1B and 5-HT1D receptors expressed in various mammalian cell lines. Br.J.Pharmacol. 123 1655. PMID: 9605573. Doggrellet al (1992) Further analysis of the inhibitory effects of dihydroergotamine, cyproheptadine and ketanserin on the responses of the rat aorta to 5-hydroxytryptamine. J.Auton.Pharmacol. 12 223. PMID: 1512277. Villalonet al (1992) Effects of S9977 and dihydroergotamine in an animal experimental model for migraine. Pharmacol.Res. 25 125. PMID: 1635891. de Boeret al (1991) Carotid vascular effects of ergotamine and dihydroergotamine in the pig: no exclusive mediation via 5-HT1-like receptors. Br.J.Pharmacol. 104 183. PMID: 1664762. |