货号 | 0454/100 |
别名 | 1-Phenylcyclopentanecarboxylic acid 2-(2-diethylaminoethoxy)ethyl ester citrate; Pentoxyverine citrate |
供应商 | Tocris |
生物活性 | A selective ligand for the σ1-site. |
运输条件 | Blue Ice |
存放说明 | Ambient |
纯度 | >99 % |
计算分子量 | 525.59 |
分子式 | C20H31NO3.C6H8O7 |
可溶性/溶解性 | Soluble to 75 mM in DMSO |
CAS号 | 23142-01-0 |
参考文献 | Quirionet al (1992) A proposal for the classification of sigma binding sites. TiPS 13 85. PMID: 1315463. Rothmanet al (1991) Labelling by [3H]1,3-di(2-tolyl)guanidine of two high affinity binding sites in guinea pig brain: evidence for allosteric regulation by calcium channel antagonists and pseudoallosteric modulation by σ ligands. Mol.Pharmacol. 39 222. PMID: 1847495. |