| 货号 | 0623/100 |
| 别名 | 1-(4-Amino-6,7-dimethoxy-2-quinazol |
| 供应商 | Tocris |
| 生物活性 | α1andα2B-adrenoceptor antagonist. Also a potent antagonist at the melatonin MT3 receptor (Ki = 10.2 nM). Also available as part of the α1-Adrenoceptor Tocriset™ and Mixed Adrenergic Tocriset™. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >99 % |
| 计算分子量 | 419.87 |
| 分子式 | C19H21N5O4.HCl |
| 可溶性/溶解性 | Soluble to 25 mM in DMSO and to 5 mM in ethanol |
| CAS号 | 19237-84-4 |
| 参考文献 | Paulet al (1999) Characterisation of 2-[125I]iodomelatonin binding sites in syrian hamster peripheral organs. J.Pharmacol.Exp.Ther. 290 334. PMID: 10381796. Matheet al (1996) Prazosin inhibits MK-801-induced hyperlocomotion and dopamine release in the nucleus accumbens. Eur.J.Pharmacol. 309 1. PMID: 8864686. Pickering and Niles (1990) Pharmacological characterization of melatonin binding sites in Syrian hamster hypothalamus. Eur.J.Pharmacol. 175 71. PMID: 2157597. Merck Index 127897. |