| 货号 | 4591/1 |
| 供应商 | Tocris |
| 生物活性 | Potentδ-opioid receptor agonist (IC50 = 0.5 nM in human granulocytes). Exhibits a high rate of blood-brain barrier penetrance. |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 计算分子量 | 768.87 |
| 分子式 | C37H52N8O10< |
| 可溶性/溶解性 | Soluble to 0.40 mg/ml in 50% acetonitrile / water |
| 序列号 | YAFDVVG (Modifications: Ala-2 = D-Ala, Gly-7 = C-terminal amide) |
| 参考文献 | Fioriet al (1997) Deltorphin transport across the blood-brain barrier. Proc.Natl.Acad.Sci.USA 94 9469. PMID: 9256506. Stefanoet al (1992) [D-Ala2]Deltorphin I binding and pharmacological evidence for a special subtype of δ opioid receptor on human and invertebrate immune cells. Proc.Natl.Acad.Sci.USA 89 9316. PMID: 1329092. Erspameret al (1989) Deltorphins: a family of naturally occurring peptides with high affinity and selectivity for δ opioid binding sites. Proc.Natl.Acad.Sci.USA 86 5188. PMID: 2544892. |