| 货号 | 1709/10 |
| 别名 | 3-Methyl-6-[-3-(trifluoromethyl)phe |
| 供应商 | Tocris |
| 生物活性 | Benzodiazepine agonist displaying selectivity for α1 subunit-containing GABAA receptors (Ki values are 130, 1820, 1530, > 10000, 490 and > 10000 nM for α1,α2,α3,α4,α5 and α6-subunit containing receptors respectively). Orally active anxiolytic and anticonvulsant in vivo. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >99 % |
| 计算分子量 | 278.24 |
| 分子式 | C13H9F3N4 |
| 可溶性/溶解性 | Soluble to 50 mM in DMSO and to 25 mM in ethanol |
| CAS号 | 66548-69-4 |
| 参考文献 | Sieghart (1995) Structure and pharmacology of γ-aminobutyric acidA receptor subtypes. Pharmacol.Rev. 47 181. PMID: 7568326. Lippaet al (1979) Benzodiazepine receptors: cellular and behavioral characteristics. Pharmacol.Biochem.Behav. 10 831. PMID: 40258. Squireset al (1979) Some properties of brain specific benzodiazepine receptors: new evidence for multiple receptors. Pharmacol.Biochem.Behav. 10 825. PMID: 40257. |