| 货号 | 2924/50 |
| 别名 | 6-S-[(4-Nitrophenyl)methyl]-6-thioi |
| 供应商 | Tocris |
| 生物活性 | Equilibrative nucleoside transporter 1 (ENT1) inhibitor (Ki values are 0.4 and 2800 nM for hENT1 and hENT2 respectively). |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >99 % |
| 计算分子量 | 419.41 |
| 分子式 | C17H17N5O6S |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO |
| CAS号 | 38048-32-7 |
| 参考文献 | Lin and Buolamwini (2007) Synthesis and flow cytometric evaluation, and identification of highly potent dipyridamole analogues as equilibrative nucleoside transporter 1 inhibitors. J.Med.Chem. 50 3906. PMID: 17636949. Tsujieet al (2007) Human equilibrative nucleoside transporter 1, as a predictor of 5-fluorouracil resistance in human pancreatic cancer. Anticancer Res. 27 2241. PMID: 17695509. Wardet al (2000) Kinetic and pharmacological properties of cloned human equilibrative nucleoside transporters, ENT1 and ENT2, stably expressed in nucleoside transporter-deficient PK15 cells. J.Biol.Chem. 275 8375. PMID: 10722669. |