货号 | 3227/1 |
别名 | Kallidin |
供应商 | Tocris |
生物活性 | Endogenous bradykinin receptor agonist that displays some selectivity for the B2 receptor (Ki values are 2.54 and 0.63 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces peripheral vascular resistance in vivo. Twice as potent as bradykinin (Cat No. 3004) in vivo. |
运输条件 | Blue Ice |
存放说明 | -20℃ |
计算分子量 | 1188.39 |
分子式 | C56H85N17O12 |
可溶性/溶解性 | Soluble to 5 mg/ml in water |
CAS号 | 342-10-9 |
序列号 | KRPPGFSPFR |
参考文献 | Leeb-Lundberget al (2005) International union of pharmacology. XLV. Classification of the kinin receptor family: from molecular mechanisms to pathophysiological consequences. Pharmacol.Rev. 57 27. PMID: 15734727. Regoliet al (2001) Classification of kinin receptors. Biol.Chem. 382 31. PMID: 11258668. Regoli and Barabe (1980) Pharmacology of bradykinin and related kinins. Pharmacol.Rev. 32 1. PMID: 7015371. |