| 货号 | 3225/1 |
| 别名 | Des-Arg10-Kallidin |
| 供应商 | Tocris |
| 生物活性 | Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2 receptors respectively). Hypotensive agent that reduces peripheral vascular resistance in vivo. 16-fold more potent than [Des-Arg9]-Bradykinin (Cat No. 3005). |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 计算分子量 | 1032.21 |
| 分子式 | C50H73N13O11 |
| 可溶性/溶解性 | Soluble to 1 mg/ml in water |
| CAS号 | 71800-36-7 |
| 序列号 | KRPPGFSPF |
| 参考文献 | Leeb-Lundberget al (2005) International union of pharmacology. LV. Classification of the kinin receptor family: from molecular mechanisms to pathophysiological consequences. Pharmacol.Rev. 57 27. PMID: 15734727. Regoliet al (2001) Classification of kinin receptors. Biol.Chem. 382 31. PMID: 11258668. Drapeauet al (1991) Hypotensive effects of Lys-des-Arg9-Bradykinin and metabolically protected agonists of B1 receptors for kinins. J.Pharmacol.Exp.Ther. 259 997. PMID: 1662280. |