| 货号 | 1955/10 |
| 别名 | 6-[2-[4-[Bis(4-fluorophenyl)methyle |
| 供应商 | Tocris |
| 生物活性 | Potent and long-acting 5-HT2 receptor antagonist (Ki = 0.39 nM). Anxiolytic in vivo. |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >99 % |
| 计算分子量 | 477.57 |
| 分子式 | C27H25F2N3OS |
| 可溶性/溶解性 | Soluble to 25 mM in ethanol and to 100 mM in DMSO |
| CAS号 | 87051-43-2 |
| 参考文献 | Watanabeet al (1992) Syntheses and 5-HT2 antagonist activity of bicyclic 1,2,4-triazol-3(2H)-one and 1,3,5-triazine-2,4(3H)-dione derivatives. J.Med.Chem. 35 189. PMID: 1732528. Janssen (1985) Pharmacology of potent and selective S2-serotonergic antagonists. J.Cardiovasc.Pharmacol. 7 S2. PMID: 2412048. Leysenet al (1985) Receptor-binding properties in vitroandin vivo of ritanserin. Mol.Pharmacol. 27 600. PMID: 2860558. |