| 货号 | 0590/10 |
| 别名 | [(8β)-1,6-Dimethylergolin-8-yl)methy |
| 供应商 | Tocris |
| 生物活性 | Antagonist at 5-HT1/5-HT2 with activity at 5-HT1D. Has moderate affinity for 5-HT6 and high affinity for 5-HT7. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 计算分子量 | 403.52 |
| 分子式 | C25H29N3O2 |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO |
| CAS号 | 17692-51-2 |
| 参考文献 | Aulakhet al (1992) Effects of various serotonin receptor subtype selective antagonists alone and on m-chlorophenylpiperazine-induced neuroendocrine changes in rats. J.Pharmacol.Exp.Ther. 263 588. PMID: 1432690. Bagdyet al (1992) Pharmacological characterization of serotonin receptor subtypes involved in vasopressin and plasma renin activity responses to serotonin agonists. Eur.J.Pharmacol. 210 285. PMID: 1535317. Milleret al (1992) Agonist activity of sumatriptan and metergoline at the human 5-HT1Dβ receptor in the action of sumatriptan. Eur.J.Pharmacol. 227 99. PMID: 1330643. |