| 货号 | 0514/10 |
| 别名 | 1-(2-Diphenylmethoxyethyl)-4-(3-phe |
| 供应商 | Tocris |
| 生物活性 | Potent and selective inhibitor of dopamine uptake (KD = 5.5 nM in rat striatal membranes). |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 计算分子量 | 487.51 |
| 分子式 | C28H34N2O.2HCl |
| 可溶性/溶解性 | Soluble to 5 mM in DMSO |
| CAS号 | 76778-22-8 |
| 参考文献 | Reithet al (1994) GBR 12909 and 12935 block dopamine uptake into brain synaptic vesicles as well as nerve endings. Eur.J.Pharmacol. 253 175. PMID: 8013544. Reithet al (1992) Evidence for mutually exclusive binding of cocaine, BTCP, GBR 12935, and dopamine to the dopamine transporter. Eur.J.Pharmacol. 227 417. PMID: 1446712. Andersenet al (1987) Biochemical and pharmacological characterization of [3H]GBR 12935 binding in vitro to rat striatal membranes: labelling of the dopamine uptake complex. J.Neurochem. 48 1887. PMID: 2952763. |