| 货号 | 2710/1 |
| 别名 | 2-[4-[[3-(4-Bromophenyl)-1-oxo-2-pr |
| 供应商 | Tocris |
| 生物活性 | Heparanase inhibitor (IC50 = 0.4 μM) that displays no major inhibition of human cytochrome P450 isoenzymes (IC50 > 30 μM). Exhibits antiangiogenic properties in vitro(IC50 = 1 μM). |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >98 % |
| 计算分子量 | 495.3 |
| 分子式 | C24H16BrFN2O4 |
| 可溶性/溶解性 | Soluble to 10 mM in DMSO |
| CAS号 | 853929-59-6 |
| 参考文献 | McKenzie (2007) Heparanase: a target for drug discovery in cancer and inflammation. Br.J.Pharmacol. 151 1. PMID: 17339837. Courtneyet al (2005) Furanyl-1,3-thiazol-2-yl and benzoxazol-5-yl acetic acid derivates: novel classes of heparanase inhibitor. Bioorg.Med.Chem.Letts. 152295. |