货号 | 1691/10 |
别名 | 1-(6-Amino-9H-purin-9-yl)-1-deoxy-N |
供应商 | Tocris |
生物活性 | High affinity adenosine receptor agonist (Ki values are 6.2, 14, and 20 nM for human A3, A1 and A2A receptors respectively; EC50 = 2.4 μM for human A2B). Inhibits platelet aggregation and is centrally active in vivo. |
运输条件 | Blue Ice |
存放说明 | 4℃ |
纯度 | >99 % |
计算分子量 | 308.3 |
分子式 | C12H16N6O4 |
可溶性/溶解性 | Soluble to 40 mM in DMSO |
CAS号 | 35920-39-9 |
参考文献 | Knappet al (2001) Adenosine agonists CGS21680 and NECA inhibit the initiation of cocaine self-administration. Pharmacol.Biochem.Behav. 68 797. PMID: 11526979. Klotz (2000) Adenosine receptors and their ligands. Naunyn Schmiedebergs Arch.Pharmacol. 362 382. PMID: 11111832. Cusack and Hourani (1981) 5'-N-ethylcarboxamidoadenosine: a potent inhibitor of human platelet aggregation. Br.J.Pharmacol. 72 443. PMID: 7260485. |