| 货号 | 0206/1G |
| 供应商 | Tocris |
| 生物活性 | Non-specific endogenous agonist at the inhibitory glycine receptor. More selective than taurine (Cat. No. 0209). Also distinguishes between GABA transporters (IC50 values are 19, 58, 110, 1320 and 5690 μM for rGAT-2, hGAT-3, rGAT-3, hBGT-3 and hGAT-1 respectively). |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 计算分子量 | 89.09 |
| 分子式 | C3H7NO2 |
| 可溶性/溶解性 | Soluble to 100 mM in water |
| 参考文献 | Schieden and Betz (1995) Pharmacology of the inhibitory glycine receptor: agonist and antagonist actions of amino acids and piperidine carboxylic acid compounds. Mol.Pharmacol. 48 919. PMID: 7476923. Bordenet al (1994) Tiagabine, SK&F 89976-A, CI 966, and NNC-711 are selective for the cloned GABA transporter GAT-1. Eur.J.Pharmacol. 269 219. PMID: 7851497. Saitohet al (1994) A novel antagonist, phenylbenzene ω-phosphono-α-amino acid, for strychnine-sensitive glycine receptors in the rat spinal cord. Br.J.Pharmacol. 113 165. PMID: 7812607. |