JTC 801
货号：
21254-5mg 基本售价：
630.0 元 规格：
5 mg
产品信息
概述| 货号 | 21254-5mg |
| 描述 | JTC 801 is an antagonist of the nociceptin receptor (ORL1; Ki = 44.5 nM; IC50 = 94 nM) that is >100-, >100-, and >3-fold more selective for ORL1 over the related δ-, κ-, and µ-opioid receptors, respectively.1 It demonstrates anti-nociceptive effects in acute pain models in mice upon oral administration at 1 mg/kg.1 |
性能| 供应商 | Cayman |
| 应用文献 |
1.Yamada, H.,Nakamoto, H.,Suzuki, Y., et al. Pharmacological profiles of a novel opioid receptor-like1 (ORL(1)) receptor antagonist, JTC-801. Br. J. Pharmacol. 135(2), 323-332 (2002).
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| 运输条件 | Wet ice in continental US; may vary elsewhere |
| 存放说明 | -20 |
| 纯度 | ≥98% |
| 计算分子量 | 448 |
| 分子式 | C26H25N3O2 • HCl |
| CAS号 | 244218-51-7 |
| 稳定性 | ≥ 2 years |
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