Blonanserin
货号：
16480-5mg 基本售价：
490.0 元 规格：
5 mg
产品信息
概述| 货号 | 16480-5mg |
| 描述 | Blonanserin is a 4-phenyl-2-(1-piperazinyl) pyridine that acts as an antagonist at dopamine D2, D3, and serotonin 5-HT2A receptors (Kis = 0.14, 0.49, and 0.81 nM, respectively).1 It binds to 5-HT6 with a Ki value of 11.7 nM and demonstrates relatively low affinity for 5-HT2C(Ki = 26.4 nM), adrenergic α1(Ki = 26.7 nM), histamine H1(Ki = 765 nM), and muscarinic M1 receptors (Ki = 100 nM).1 Blonanserin was developed in Japan as a novel antipsychotic that displays 20- and 94-fold higher affinity for D2 receptors compared to haloperidol (Item No. 12014) and risperidone (Item No. 13629), respectively.1 |
| 别名 | AD5423;Lonasen; |
性能| 供应商 | Cayman |
| 应用文献 |
1.Tenjin, T.,Miyamoto, S.,Ninomiya, Y., et al. Profile of blonanserin for the treatment of schizophrenia. Neuropsychiatric Disease and Treatment 9, 587-594 (2013).
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| 运输条件 | Room temperature in continental US; may vary elsewhere |
| 存放说明 | -20 |
| 纯度 | ≥98% |
| 计算分子量 | 367.5 |
| 分子式 | C23H30FN3 |
| CAS号 | 132810-10-7 |
| 稳定性 | ≥ 2 years |
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