CGP 36216 (hydrochloride)
货号：
11985-1mg 基本售价：
490.0 元 规格：
1 mg
产品信息
概述| 货号 | 11985-1mg |
| 描述 | CGP 36216 is a selective antagonist of GABAB receptors (IC50 = 43 µM).1,2 Its action is reversed by the GABAB receptor agonist baclofen.2 It is active at presynaptic, but not postsynaptic, receptors.2 |
性能| 供应商 | Cayman |
| 应用文献 |
1.Froestl, W.,Mickel, S.J.,von Sprecher, G., et al. Phosphinic acid analogues of GABA. 2. Selective, orally active GABAB antagonists. Journal of Medicinal Chemistry 38, 3313-3331 (1995).
2.Ong, J.,Bexis, S.,Marino, V., et al. CGP 36216 is a selective antagonist at GABAB presynaptic receptors in rat brain. European Journal of Pharmacology 415, 191-195 (2001).
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| 运输条件 | Wet ice in continental US; may vary elsewhere |
| 存放说明 | -20 |
| 纯度 | ≥98% |
| 计算分子量 | 187.6 |
| 分子式 | C5H14NO2P • HCl |
| CAS号 | 1781834-71-6 |
| 稳定性 | ≥ 2 years |
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