Leelamine (hydrochloride)
货号：
10008614-5mg 基本售价：
490.0 元 规格：
5 mg
产品信息
概述| 货号 | 10008614-5mg |
| 描述 | Leelamine is a diterpene molecule whose name derives from the Sanskrit word leela which means “play”. It has weak affinity for the human central cannabinoid (CB1) and peripheral cannabinoid (CB2) receptors, exhibiting 20% displacement of [3H]-CP55940 at a concentration of 10 µM.1 Leelamine inhibits pyruvate dehydrogenase kinase (PDK) with an IC50 of 9.5 µM.2 Derivatives of leelamine exhibit anti-inflammatory activity and show moderate inhibition of phospholipase A2 activity from a variety of sources.3 |
| 别名 | Dehydroabietylamine; |
性能| 供应商 | Cayman |
| 应用文献 |
1.Martin, B.R. Leelamine. (2006).
2.Aicher, T.D.,Damon, R.E.,Koletar, J., et al. Triterpene and diterpene inhibitors of pyruvate dehydrogenase kinase (PDK). Bioorganic & Medicinal Chemistry Letters 9, 2223-2228 (1999).
3.Wilkerson, W.,DeLucca, I.,Galbraith, W., et al. Antiinflammatory phospholipase-A2 inhibitors. I. European Journal of Medicinal Chemistry 26, 667-676 (1991).
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| 运输条件 | Room temperature in continental US; may vary elsewhere |
| 存放说明 | -20 |
| 纯度 | ≥98% |
| 计算分子量 | 321.9 |
| 分子式 | C20H31N • HCl |
| CAS号 | 16496-99-4 |
| 稳定性 | ≥ 2 years |
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