S-ethyl N-[4-(trifluoromethyl)phenyl] Isothiourea (hydrochloride)
货号：
81280-5mg 基本售价：
350.0 元 规格：
5 mg
产品信息
概述| 货号 | 81280-5mg |
| 描述 | EPIT is a selective, competitive inhibitor of nNOS having a Ki of 0.32 µM for the purified human enzyme. EPIT exhibits 115-fold and 29-fold selectivity for nNOS compared to iNOS and eNOS, respectively. It exhibits reduced inhibitory potency in whole-cell assays, possibly due to reduced intracellular uptake.1 |
| 别名 | EPIT; |
性能| 供应商 | Cayman |
| 应用文献 |
1.Shearer, B.G.,Lee, S.,Oplinger, J.A., et al. Substituted N-phenylisothioureas: Potent inhibitors of human nitric oxide synthase with neuronal isoform selectivity. Journal of Medicinal Chemistry 40, 1901-1905 (1997).
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| 运输条件 | Wet ice in continental US; may vary elsewhere |
| 存放说明 | -20 |
| 纯度 | ≥98% |
| 计算分子量 | 284.7 |
| 分子式 | C10H11F3N2S • HCl |
| CAS号 | 163490-78-6 |
| 稳定性 | ≥ 1 year |
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