Eltoprazine (hydrochloride)
货号：
18428-1mg 基本售价：
350.0 元 规格：
1 mg
产品信息
概述| 货号 | 18428-1mg |
| 描述 | Eltoprazine is a phenylpiperazine compound that acts as a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Kis = 40, 52, and 81 nM, respectively).1 It exerts a dose-dependent decrease in aggressive behavior in resident-intruder tests with rats (ID50 = 0.24 mg/kg).2 |
| 别名 | DU-28,853;DU-28,893; |
性能| 供应商 | Cayman |
| 应用文献 |
1.Schipper, J.,Tulp, M.T., and Sijbesma, H. Neurochemical profile of eltoprazine. Drug Metabol.Drug Interact. 8(102), 85-114 (1990).
2.de Boer, S.F.,Lesourd, M.,Mocaer, E., et al. Selective antiaggressive effects of alnespirone in resident-intruder test are mediated via 5-hydroxytryptamine1A receptors: A comparative pharmacological study with 8-hydroxy-2-dipropylaminotetralin, ipsapirone, buspirone, eltoprazine, and WAY-100635. Journal of Pharmacology and Experimental Therapeutics 288(3), 1125-1133 (1999).
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| 运输条件 | Room temperature in continental US; may vary elsewhere |
| 存放说明 | -20 |
| 纯度 | ≥98% |
| 计算分子量 | 256.7 |
| 分子式 | C12H16N2O2 • HCl |
| CAS号 | 98206-09-8 |
| 稳定性 | ≥ 2 years |
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