GSK264220A
货号：
13009-1mg 基本售价：
350.0 元 规格：
1 mg
产品信息
概述| 货号 | 13009-1mg |
| 描述 | Endothelial lipase, a member of the triglyceride lipase gene family expressed in endothelial cells, prefers phospholipid-enriched high-density lipoprotein (HDL) over triglyceride as substrate. GSK264220A is a potent inhibitor of endothelial lipase (IC50 = 16 nM).1 Levels of HDL cholesterol are inversely correlated with endothelial lipase protein activity. Therefore, inhibition of endothelial lipase by compounds like GSK264220A may be expected to increase HDL levels and potentially decrease the risk of cardiovascular disease. |
性能| 供应商 | Cayman |
| 应用文献 |
1.Keller, P.M.,Rust, T.,Murphy, D.J., et al. A high-throughput screen for endothelial lipase using HDL as substrate. Journal of Biomolecular Screening 13(6), 468-475 (2008).
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| 运输条件 | Room temperature in continental US; may vary elsewhere |
| 存放说明 | -20 |
| 纯度 | ≥98% |
| 计算分子量 | 363.4 |
| 分子式 | C17H21N3O4S |
| CAS号 | 685506-42-7 |
| 稳定性 | ≥ 2 years |
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