CAY10570
货号:
10010032-500ug 基本售价:
322.0 元 规格:
500 ug
产品信息
概述货号 | 10010032-500ug |
描述 | The enzyme fatty acid amide hydrolase (FAAH) is capable of hydrolyzing and inactivating anandamide and other fatty acid amides that act as agonists for the central cannabinoid (CB1) receptor.1 CAY10570 is a reversible competitive inhibitor of FAAH activity exhibiting an IC50 value of 1.3 µM.2 CAY10570 has no affinity for the human CB1 receptor and acts as a competitive inhibitor of FAAH activity without being hydrolyzed by the enzyme.2 |
性能供应商 | Cayman |
应用文献 |
1.Cravatt, B.F.,Giang, D.K.,Mayfield, S.P., et al. Molecular characterization of an enzyme that degrades neuromodulatory fatty-acid amides. Nature 384, 83-87 (1996). 2.Muccioli, G.G.,Fazio, N.,Scriba, G.K.E., et al. Substituted 2-thioxoimidazolidin-4-ones and imidazolidine-2,4-diones as fatty acid amide hydrolase inhibitors templates. Journal of Medicinal Chemistry 49, 417-425 (2006).
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运输条件 | Room temperature in continental US; may vary elsewhere |
存放说明 | -20 |
纯度 | >98% |
计算分子量 | 408.6 |
分子式 | C25H32N2OS |
CAS号 | 875014-22-5 |
稳定性 | ≥ 1 year |
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